Cyproterone acetate wikipedia
WebUses. Cyproterone is used for reducing male hypersexuality, and in prostatic cancer and severe female hirsutism. A formulation of cyproterone plus ethinylestradiol (Dianette, which contains only 2 mg of cyproterone acetate) is offered for this latter purpose as well as for severe acne in women; this preparation acts as an oral contraceptive but does not have … WebNPS MedicineWise
Cyproterone acetate wikipedia
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Cyproterone acetate (CPA), sold alone under the brand name Androcur or with ethinylestradiol under the brand names Diane or Diane-35 among others, is an antiandrogen and progestin medication used in the treatment of androgen-dependent conditions such as acne, excessive body hair … See more CPA is used as a progestin and antiandrogen in hormonal birth control and in the treatment of androgen-dependent conditions. Specifically, CPA is used in combined birth control pills, in the treatment of … See more CPA is generally well-tolerated and has a mild side-effect profile regardless of dosage when it is used in combination with an estrogen in women. Side effects of CPA in general include hypogonadism (low sex-hormone levels) and associated symptoms such as See more Inhibitors and inducers of the cytochrome P450 enzyme CYP3A4 may interact with CPA. Examples of strong CYP3A4 inhibitors include See more CPA, also known as 1α,2α-methylene-6-chloro-17α-acetoxy-δ -progesterone or as 1α,2α-methylene-6-chloro-17α-hydroxypregna-4,6-diene-3,20-dione acetate, is a synthetic pregnane steroid and an acetylated derivative of 17α-hydroxyprogesterone. … See more Contraindications of CPA include: • Hypersensitivity to CPA or any of the other components of the medication • Pregnancy, lactation, and breastfeeding • Puberty (except if being used to treat precocious puberty or delay puberty) See more CPA is relatively safe in acute overdose. It is used at very high doses of up to 300 mg/day by mouth and 700 mg per week by intramuscular … See more Pharmacodynamics CPA has antiandrogenic activity, progestogenic activity, weak partial glucocorticoid activity, weak steroidogenesis inhibitor activity, and agonist activity at the pregnane X receptor. It has no See more WebHot flushes and sweats. Hot flushes are a common side effect of this treatment. During a flush, your neck and face may feel warm and look red. Flushes may last from a few seconds up to 10 minutes. You may have sweats and then feel cold and clammy. Some people feel anxious or irritable during a hot flush.
WebCyproterone acetate is metabolized by the CYP3A4 enzyme, forming the active metabolite 15β-hydroxycyproterone acetate, which retains its antiandrogen activity, but has reduced …
WebThe side effects of cyproterone acetate (CPA), a steroidal antiandrogen and progestin, including its frequent and rare side effects, have been studied and characterized.It is generally well-tolerated and has a mild side-effect profile, regardless of dosage, when it used as a progestin or antiandrogen in combination with an estrogen such as … WebDrug information provided by: IBM Micromedex At first, cyproterone often causes loss of strength and energy or tiredness. However, these effects are lessened after about the third month of treatment and it is very important that you continue to receive this medication.
The pharmacology of cyproterone acetate (CPA) concerns the pharmacology (pharmacodynamics, pharmacokinetics, and routes of administration) of the steroidal antiandrogen and progestin medication cyproterone acetate. CPA blocks the effects of androgens like testosterone in the body, which it does by preventing them from interacting with their biological target, the androgen re…
Webcyproterone acetate ( uncountable ) ( organic chemistry, pharmacology) The cyproterone ester of acetic acid that is an antiandrogen and progestin medication - C 24 H 29 ClO 4. … litter of chihuahua puppiesWebCyproterone acetate has been associated with an overall rare, but cumulative dose-dependent, increased risk of meningioma (single and multiple), mainly at doses of 25 … litter of 24 puppiesWebCyproterone acetate and testosterone levels with 300 mg per week cyproterone acetate by intramuscular injection in men.png 1,825 × 1,103; 292 KB Cyproterone acetate … litter of bunnies calledWebCyproterone, also known by its developmental code name SH-80881, is a steroidal antiandrogen which was studied in the 1960s and 1970s but was never introduced for medical use.[1][2][3] It is an analogue of cyproterone acetate , an antiandrogen, progestin, and antigonadotropin which was introduced instead of cyproterone and is widely used … litter of cats is calledWebcyproterone acetate is diagnosed with meningioma, treatment with cyproterone acetate must be stopped (see section 4.3). Diabetes . Strict medical supervision is necessary if the patient suffers from diabetes, because the requirement for oral antidiabetics or insulin can change during treatment cyproterone acetate (see section 4.3). litter of catsWebOct 24, 2024 · File:Cyproterone acetate.svg From Wikimedia Commons, the free media repository Jump to navigation Jump to search File File history File usage on Commons … litter of cubsWebWhat will it do for me? This medication contains a combination of two ingredients: cyproterone and ethinyl estradiol. Cyproterone belongs to a group of medications known as antiandrogens. Ethinyl estradiol belongs to a group of medications known as estrogens. litter of dogs meaning